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STRUCTURE OF RET PROTEIN TYROSINE KINASE DOMAIN IN COMPLEX WITH NINTEDANIB

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Protein Data Bank Japan2023-10-11 更新2026-03-21 收录
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STRUCTURE OF RET PROTEIN TYROSINE KINASE DOMAIN IN COMPLEX WITH NINTEDANIB Descriptor: FORMIC ACID, Proto-oncogene tyrosine-protein kinase receptor Ret, methyl (3Z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1H-indole-6-carboxylate Authors: Terzyan, S.S, Shen, T, Wu, J, Mooers, B.H.M. Deposit date: 2018-12-17 Release date: 2019-06-05 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (1.87 Å) Cite: Structural basis of resistance of mutant RET protein-tyrosine kinase to its inhibitors nintedanib and vandetanib. J.Biol.Chem., 294, 2019

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2018-12-17
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