Palladium-Catalyzed Sequential Vinylic C–H Arylation/Amination of 2‑Vinylanilines with Aryl boronic Acids: Access to 2‑Arylindoles
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A palladium-catalyzed selective and successive vinylic C–H arylation/amination of 2-vinylanilines with arylboronic acids to generate indoles has been developed. This procedure represents a straightforward and practical approach to valuable multifunctionalized indoles.
创建时间:
2017-12-08



