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PPARgamma ligand-binding domain in complex with PG08-NL

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Protein Data Bank Japan2025-12-03 更新2026-04-19 收录
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PPARgamma ligand-binding domain in complex with PG08-NL Descriptor: DI(HYDROXYETHYL)ETHER, PG08-NL, Peroxisome proliferator-activated receptor gamma Authors: Sigal, M, Okada, C, Katoh, T, Suga, H, Sengoku, T. Deposit date: 2025-05-29 Release date: 2025-11-05 Last modified: 2025-12-03 Method: X-RAY DIFFRACTION (1.39 Å) Cite: De Novo Discovery of alpha , alpha-Disubstituted alpha-amino Acid-Containing alpha-helical Peptides as Competitive PPAR gamma PPI Inhibitors. J.Am.Chem.Soc., 147, 2025

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2025-05-29
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