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Crystal Structure of Human Pirin in complex with a Chemical Probe pyrrolidine 24

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Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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Crystal Structure of Human Pirin in complex with a Chemical Probe pyrrolidine 24 Descriptor: DIMETHYL SULFOXIDE, FE (III) ION, GLYCEROL, ... Authors: Ali, S, van Montfort, R. Deposit date: 2016-04-15 Release date: 2017-01-11 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (1.73 Å) Cite: Discovery of a Chemical Probe Bisamide (CCT251236): An Orally Bioavailable Efficacious Pirin Ligand from a Heat Shock Transcription Factor 1 (HSF1) Phenotypic Screen. J. Med. Chem., 60, 2017

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2016-04-15
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