遇见数据集

JAK2 JH1 in complex with PN3-115

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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JAK2 JH1 in complex with PN3-115 Descriptor: 2-{5-[(2-{[3,5-difluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-5-methylpyrimidin-4-yl)amino]-2-fluorophenyl}-1lambda~6~,2-thiazolidine-1,1-dione, Tyrosine-protein kinase JAK2 Authors: Davis, R.R, Schonbrunn, E. Deposit date: 2020-01-29 Release date: 2021-02-17 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Structural Insights into JAK2 Inhibition by Ruxolitinib, Fedratinib, and Derivatives Thereof. J.Med.Chem., 64, 2021

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2020-01-29
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