遇见数据集

USP7 IN COMPLEX WITH LIGAND COMPOUND 1

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Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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USP7 IN COMPLEX WITH LIGAND COMPOUND 1 Descriptor: 3-({4-hydroxy-1-[(2R)-2-methyl-3-phenylpropanoyl]piperidin-4-yl}methyl)quinazolin-4(3H)-one, Ubiquitin carboxyl-terminal hydrolase 7 Authors: Leger, P.R, Wustrow, D.J, Hu, D.X, Krapp, S, Maskos, K, Blaesse, M. Deposit date: 2020-01-29 Release date: 2020-04-29 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.69 Å) Cite: Discovery of Potent, Selective, and Orally Bioavailable Inhibitors of USP7 with In Vivo Antitumor Activity. J.Med.Chem., 63, 2020

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2020-01-29
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