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JAK2 JH2 in complex with JAK179

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Protein Data Bank Japan2023-10-11 更新2026-03-21 收录
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JAK2 JH2 in complex with JAK179 Descriptor: GLYCEROL, Tyrosine-protein kinase JAK2, [4-({5-amino-3-[(4-sulfamoylphenyl)amino]-1H-1,2,4-triazole-1-carbonyl}amino)phenoxy]acetic acid Authors: Krimmer, S.G, Liosi, M.E, Schlessinger, J, Jorgensen, W.L. Deposit date: 2019-03-20 Release date: 2020-03-25 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (1.71 Å) Cite: Selective Janus Kinase 2 (JAK2) Pseudokinase Ligands with a Diaminotriazole Core. J.Med.Chem., 63, 2020

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2019-03-20
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