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Structure of spastin AAA domain in complex with a quinazoline-based inhibitor

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Protein Data Bank Japan2023-10-11 更新2026-03-21 收录
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Structure of spastin AAA domain in complex with a quinazoline-based inhibitor Descriptor: (4S)-2-METHYL-2,4-PENTANEDIOL, N-(3-tert-butyl-1H-pyrazol-5-yl)-2-[(2R)-2-methylpiperazin-1-yl]quinazolin-4-amine, SULFATE ION, ... Authors: Pisa, R, Cupido, T, Kapoor, T.M. Deposit date: 2019-02-12 Release date: 2019-03-27 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (2.425 Å) Cite: Designing Allele-Specific Inhibitors of Spastin, a Microtubule-Severing AAA Protein. J. Am. Chem. Soc., 141, 2019

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2019-02-12
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