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Crystal structure of human CLK1 in complex with Leucettinib-21

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Protein Data Bank Japan2024-07-31 更新2026-04-19 收录
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Crystal structure of human CLK1 in complex with Leucettinib-21 Descriptor: (4~{Z})-4-(1,3-benzothiazol-6-ylmethylidene)-2-[[(2~{R})-1-methoxy-4-methyl-pentan-2-yl]amino]-1~{H}-imidazol-5-one, Dual specificity protein kinase CLK1 Authors: Kraemer, A, Schroeder, M, Meijer, L, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2023-05-09 Release date: 2023-05-17 Last modified: 2024-07-31 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Chemical, Biochemical, Cellular, and Physiological Characterization of Leucettinib-21, a Down Syndrome and Alzheimer's Disease Drug Candidate. J.Med.Chem., 66, 2023

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2023-05-09
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