遇见数据集

Tankyrase 2 in complex with an inhibitor (OUL228)

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Protein Data Bank Japan2024-01-31 更新2026-03-28 收录
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Tankyrase 2 in complex with an inhibitor (OUL228) Descriptor: 8-propan-2-yloxy-4~{H}-thieno[2,3-c]isoquinolin-5-one, GLYCEROL, Poly [ADP-ribose] polymerase tankyrase-2, ... Authors: Sowa, S.T, Lehtio, L. Deposit date: 2021-05-21 Release date: 2021-12-08 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Analogs of TIQ-A as inhibitors of human mono-ADP-ribosylating PARPs. Bioorg.Med.Chem., 52, 2021

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2021-05-21
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