Yeast 20S proteasome in complex with the vinyl sulfone LU102

Yeast 20S proteasome in complex with the vinyl sulfone LU102 Descriptor: N3Phe-Leu-Leu-Phe(4-NH2CH2)-methyl vinyl sulfone, bound form, Proteasome component C1, ... Authors: Geurink, P.P, van der Linden, W.A, Mirabella, A.C, Gallastegui, N, de Bruin, G, Blom, A.E.M, Voges, M.J, Mock, E.D, Florea, B.I, van der Marel, G.A, Driessen, C, van der Stelt, M, Groll, M, Overkleeft, H.S, Kisselev, A.F. Deposit date: 2013-01-06 Release date: 2013-01-30 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.7 Å) Cite: Incorporation of Non-natural Amino Acids Improves Cell Permeability and Potency of Specific Inhibitors of Proteasome Trypsin-like Sites. J.Med.Chem., 56, 2013