BAZ2A bromodomain in complex with compound UP39
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BAZ2A bromodomain in complex with compound UP39 Descriptor: Bromodomain adjacent to zinc finger domain protein 2A, methyl 5-[(5-ethanoyl-2-ethoxy-phenyl)carbamoyl]-2-(2-piperazin-1-ylethoxy)benzoate Authors: Dalle Vedove, A, Cazzanelli, G, Caflisch, A, Lolli, G. Deposit date: 2021-01-18 Release date: 2022-03-02 Last modified: 2025-03-26 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Reevaluation of bromodomain ligands targeting BAZ2A. Protein Sci., 32, 2023
与化合物UP39结合的BAZ2A溴结构域(bromodomain) 描述:锌指结构域旁蛋白2A(Bromodomain adjacent to zinc finger domain protein 2A,即BAZ2A),其结合配体为5-[(5-乙酰基-2-乙氧基苯基)氨基甲酰基]-2-(2-哌嗪-1-基乙氧基)苯甲酸甲酯 作者:Dalle Vedove, A、Cazzanelli, G、Caflisch, A、Lolli, G 提交日期:2021-01-18 发布日期:2022-03-02 最后修改日期:2025-03-26 实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率2.3 Å 引用:《靶向BAZ2A的溴结构域配体重评估》。《Protein Sci.》,32卷,2023年



